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original article |
Date |
Title |
Authors All Authors |
| 1 |
[GO] |
2025―Oct―30 |
Asymmetric Synthesis of MK-7845, an Investigational Treatment for COVID-19 |
Reed T. Larson, Ben W. H. Turnbull, Patrick J. Moon, Dan Lehnherr, Jonathan M. E. Hughes, Stasik Popov, et al. (+35) Gilmar A. Brito, Teresa Andreani, Suhong Kim, James Herbort, Renee J. Sifri, Shorouk O. Badir, Chibueze I. Onyeagusi, Nicholas R. Deprez, Douglas Otte, Donald R. Gauthier, Nadine Kuhl, Yining Ji, Andrew J. Neel, Ryan D. Cohen, Jeffrey S. Derrick, Cecilia Bottecchia, Clara Hartmanshenn, David A. Vargas, Guilherme Dal Poggetto, Alex M. Confer, Michelle Zheng, Yangzhong Qin, Ajit Vikram, Justin A. Newman, Zeinab Sakhaei, Riki J. Drout, Lu Chen, Zheng Wu, Steve Castro, Stella K. Betancourt, Gurpreet Longia, Brittany Kassim, Yingju Xu, Jamie M. McCabe Dunn, Nastaran Salehi Marzijarani |
| 2 |
[GO] |
2024―Jun―27 |
Synthesis of Structural ADP-Ribose Analogues as Inhibitors for SARS-CoV-2 Macrodomain 1 |
Koen J. Rijpkema, Marion Schuller, Miriam S. van der Veer, Sjoerd Rieken, Diego L. R. Chang, Pascal Balić, et al. (+8) Alex Todorov, Hugo Minnee, Sven Wijngaarden, Isaac A. Matos, Nicolas C. Hoch, Jeroen D. C. Codée, Ivan Ahel, Dmitri V. Filippov |
| 3 |
[GO] |
2023―Jul―31 |
Deuteration for Metabolic Stabilization of SARS-CoV-2 Inhibitors GC373 and Nirmatrelvir |
Tayla J. Van Oers, Alexia Piercey, Alexandr Belovodskiy, Béla Reiz, Bethan L. Donnelly, Wayne Vuong, et al. (+4) M. Joanne Lemieux, James A. Nieman, Karine Auclair, John C. Vederas |
| 4 |
[GO] |
2023―Jun―26 |
Synthetic Analogs of the Sponge Sesterterpenoid Alotaketal C are Potent Inhibitors of SARS-CoV-2 Omicron BA.1 and BA.5 Infections of Human Lung Cells |
Polina Blagojevic, Jimena Perez-Vargas, Kunzhong Jian, David E. Williams, Ivan Villanueva, Connor A. H. Thompson, et al. (+5) Siobhan Ennis, Masahiro Niikura, Ian Tietjen, François Jean, Raymond J. Andersen |
| 5 |
[GO] |
2022―Dec―07 |
A 1-Pot Synthesis of the SARS-CoV-2 Mpro Inhibitor Nirmatrelvir, the Key Ingredient in Paxlovid |
Juan C. Caravez, Karthik S. Iyer, Rahul D. Kavthe, Joseph R. A. Kincaid, Bruce H. Lipshutz |
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